Emla 5% Cream 5g Imported In Pakistan
Emla 5% Cream Overview
Emla 5% Cream is a topical anesthetic used to numb the skin before minor medical procedures. It contains a combination of lidocaine and prilocaine, both of which are effective local anesthetics.
Composition
- Active Ingredients:
- Lidocaine: 2.5g
- Prilocaine: 2.5g
- Total Volume: 5g per tube
Uses of Emla 5% Cream
Emla Cream is commonly utilized for various purposes, including:
- Numbing for Injections: Ideal for reducing pain during vaccinations or blood draws.
- Minor Surgical Procedures: Used to numb the skin prior to small surgeries.
- Tattooing: Can be applied to minimize discomfort during tattoo application (consultation with a healthcare professional is recommended).
Application Guidelines
- Timing: Apply Emla Cream at least one hour before the procedure for optimal effectiveness.
- Duration of Effect: The numbing effect typically lasts for about two hours.
Availability and Pricing in Pakistan
- Price: Approximately Rs. 9,500 for a 5g tube.
- Where to Buy: Available through various online pharmacies, including:
- Medical Mart
- Pink Pakistan
Precautions and Side Effects
Precautions
- Not Suitable For:
- Infants born before 37 weeks of gestation.
- Children under 12 years when applied to the genital area.
- Individuals with known allergies to lidocaine or prilocaine.
Possible Side Effects
- Skin irritation or allergic reactions may occur. It is advisable to consult a healthcare provider if any adverse effects are experienced.
Conclusion
Emla 5% Cream is a valuable product for those needing local anesthesia for minor procedures. Always follow application guidelines and consult with a healthcare professional if you have any concerns or specific health conditions.
Original price was: ₨5,000.00.₨3,999.00Current price is: ₨3,999.00.
Description
Emla 5% Cream Overview
Emla 5% Cream is a topical anesthetic used to numb the skin before minor medical procedures. It contains a combination of lidocaine and prilocaine, both of which are effective local anesthetics.
Composition
- Active Ingredients:
- Lidocaine: 2.5g
- Prilocaine: 2.5g
- Total Volume: 5g per tube
Uses of Emla 5% Cream
Emla Cream is commonly utilized for various purposes, including:
- Numbing for Injections: Ideal for reducing pain during vaccinations or blood draws.
- Minor Surgical Procedures: Used to numb the skin prior to small surgeries.
- Tattooing: Can be applied to minimize discomfort during tattoo application (consultation with a healthcare professional is recommended).
Application Guidelines
- Timing: Apply Emla Cream at least one hour before the procedure for optimal effectiveness.
- Duration of Effect: The numbing effect typically lasts for about two hours.
Availability and Pricing in Pakistan
- Price: Approximately Rs. 9,500 for a 5g tube.
- Where to Buy: Available through various online pharmacies, including:
- Medical Mart
- Pink Pakistan
Precautions and Side Effects
Precautions
- Not Suitable For:
- Infants born before 37 weeks of gestation.
- Children under 12 years when applied to the genital area.
- Individuals with known allergies to lidocaine or prilocaine.
Possible Side Effects
- Skin irritation or allergic reactions may occur. It is advisable to consult a healthcare provider if any adverse effects are experienced.
Conclusion
Emla 5% Cream is a valuable product for those needing local anesthesia for minor procedures. Always follow application guidelines and consult with a healthcare professional if you have any concerns or specific health conditions.
Key Benefits of Emla 5% Cream
Emla 5% Cream offers several advantages, particularly in medical and cosmetic procedures:
- Effective Pain Relief: The cream numbs the skin surface, significantly reducing pain during minor medical procedures, such as injections and skin operations.
- Dual Action: Contains two active ingredients (lidocaine and prilocaine) that work synergistically to enhance the numbing effect.
- Wide Applicability: Suitable for both adults and children, making it a versatile option for various medical situations, including vaccinations, blood donations, and minor surgeries.
- Ease of Use: Can be applied at home prior to a procedure, allowing for greater comfort and reduced anxiety, especially in children.
- Long-Lasting Effect: Provides numbness for approximately two hours, which is sufficient for most minor procedures.
Key Ingredients
Emla 5% Cream contains the following active ingredients:
- Lidocaine (2.5%): A local anesthetic that blocks nerve signals in the body, providing pain relief.
- Prilocaine (2.5%): Another local anesthetic that complements the action of lidocaine, enhancing the overall numbing effect.
Mechanism of Action
EMLA Cream (lidocaine 2.5% and prilocaine 2.5%) provides dermal analgesia (pain relief) through the following mechanism:
- When applied to intact skin under an occlusive dressing, lidocaine and prilocaine are released from the cream into the epidermal and dermal layers of the skin.
- Lidocaine and prilocaine accumulate in the vicinity of dermal pain receptors and nerve endings.
- Both lidocaine and prilocaine are amide-type local anesthetic agents that block sodium channels in the neuronal cell membranes.
- This blockade inhibits the initiation and transmission of nerve impulses, thereby preventing the sensation of pain in the treated area of the skin.
- The combination of lidocaine and prilocaine in EMLA Cream works synergistically to enhance the numbing effect compared to using either anesthetic alone.
Chemical structureSpatial arrangement of atoms in a molecule and their chemical bondsMoreDefinitionThe spatial arrangement of atoms within a molecule and the chemical bonds that hold the atoms together.ComponentsIncludes specifying the molecular geometry, electronic structure, and when necessary, the occupation of the molecule’s molecular orbitals.RepresentationRepresented using structural formulae and molecular models. Precise determination of bond lengths, angles, and torsion angles.The chemical structure of Emla Cream, which contains lidocaine and prilocaine, can be described as follows:
Lidocaine Structure
- Chemical Formula: C₁₄H₂₂N₂O
- Structural Formula:
textN
|
H2C-C-C-C-C
| | |
O N H
Lidocaine has a benzene ring connected to an amine group and an ether link, contributing to its local anesthetic properties.
Prilocaine Structure
- Chemical Formula: C₁₁H₁₅N₂O
- Structural Formula:
textN
|
H2C-C-C-C
| | |
O N H
Prilocaine is similar to lidocaine but has a slightly different structure, which also contributes to its effectiveness as a local anesthetic.
Key Precautions for Using Emla 5% Cream
- Not suitable for:
- Infants born before 37 weeks of gestation
- Children under 12 years on the genital area
- Individuals with known allergies to lidocaine, prilocaine, or any other ingredients
- Avoid contact with eyes: Can cause severe eye irritation and potential abrasion. If eye contact occurs, immediately wash out the eye with water or saline.
- Do not apply to open wounds or impaired eardrums
- Use caution in patients with severe hepatic disease: Greater risk of developing toxic plasma concentrations of lidocaine and prilocaine
- Repeated doses may increase blood levels of lidocaine and prilocaine: Use caution in acutely ill, debilitated, or elderly patients
Dietary Restrictions
There are no specific dietary restrictions mentioned in the provided search results for using Emla 5% Cream. However, it is always advisable to consult with a healthcare professional before using any medication, especially if you have any underlying health conditions or are taking other medications.
Safety During Pregnancy
- Occasional Use: According to the information available, occasional use of EMLA Cream during pregnancy is unlikely to have adverse effects on the fetus. The active ingredients, lidocaine and prilocaine, have been used by many pregnant women without serious harm reported.
- Animal Studies: Animal studies have not indicated direct or indirect harmful effects regarding pregnancy or fetal development.
- Consultation Recommended: Despite the general safety profile, it is advised that pregnant women consult their healthcare provider before using EMLA Cream to discuss potential risks and benefits.
Breastfeeding Considerations
- Excretion in Breast Milk: Both lidocaine and prilocaine can pass into breast milk, but the amounts are typically small and not considered harmful to the infant. However, breastfeeding mothers should still consult their healthcare provider before use.
Major Drug Interactions
- Antiarrhythmic Drugs:
- Examples: Tocainide, Mexiletine
- Concern: These medications can have additive effects on heart rate and rhythm, increasing the risk of cardiac complications.
- Drugs Associated with Methemoglobinemia:
- Examples:
- Nitrates/Nitrites (e.g., nitroglycerin)
- Other local anesthetics (e.g., benzocaine, bupivacaine)
- Antibiotics (e.g., dapsone, sulfonamides)
- Antineoplastic agents (e.g., cyclophosphamide)
- Concern: Concurrent use can increase the risk of methemoglobinemia, a condition where hemoglobin is altered, reducing its ability to carry oxygen.
- Examples:
- Seizure Medications:
- Examples: Phenobarbital, Phenytoin
- Concern: These may interact with the metabolic pathways of lidocaine and prilocaine.
- Other Considerations:
- Caution is advised when used with Class III antiarrhythmic drugs (e.g., amiodarone, sotalol) as specific interaction studies have not been performed.
General Recommendations
- Cumulative Doses: If using EMLA Cream in conjunction with other products containing lidocaine or prilocaine, be mindful of the total dose to avoid toxicity.
- Consult Healthcare Provider: Always inform your healthcare provider about all medications you are taking, including over-the-counter drugs and supplements, to assess potential interactions.
Dosage of Emla 5% Cream
Recommended Dosage
- Adults:
- For minor procedures (e.g., needle insertion, surgical treatment): Apply approximately 1.5 g to 2 g per 10 cm² of skin area. The cream should be applied for a minimum of 1 hour and can be left on for up to 5 hours.
- For procedures requiring deeper anesthesia (e.g., skin biopsies): Apply 1.5-2 g/10 cm² for a minimum of 2 hours.
- Children:
- Neonates (under 3 months): Apply up to 1 g on an area no larger than 10 cm².
- Infants (3-11 months): Apply up to 2 g on a total skin area no larger than 20 cm².
- Children (1-5 years): Apply up to 10 g on a skin area no larger than 100 cm².
- Children (6-11 years): Apply up to 20 g on a total skin area no larger than 200 cm².
Application Instructions
- Apply a thick layer of Emla Cream to intact skin and cover it with an airtight dressing (e.g., Tegaderm or plastic wrap) to enhance absorption.
- Ensure the cream is applied at least 1 hour before the procedure to maximize its effectiveness.
Storage
- Temperature: Store Emla Cream at temperatures between 15°C to 30°C (59°F to 86°F).
- Avoid Freezing: Do not freeze the cream.
- Shelf Life: Discard any remaining cream within 30 days after opening the tube.
Reviews
- General Feedback: Emla Cream is often praised for its effectiveness in numbing the skin before minor medical procedures. Users report a significant reduction in pain during injections and other minor surgeries.
- Ease of Use: Many appreciate the ease of application and the fact that it can be used at home before medical visits.
- Concerns: Some users have noted that the cream may not be effective for everyone, and individual experiences can vary. There are also mentions of potential side effects, such as skin irritation or allergic reactions, although these are not common.
Reviews
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